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Brand/Trademark BIOMOL

Mainfeature: TRPV1 antagonist

Target/Molecule Synonym TRPV1, FAAH
Keywords NEU/CAN| DDI/SMM Blocker| Inhibitor TRP channel| FAAH
Molecular Weight 462.7
Original Item Name N-Arachidonoyl-serotonin
Purity ≥98% (TLC)
Sample Type Pale yellow oil.
CAS Number 187947-37-1
Formula C30H42N2O2
Target TRPV1, FAAH
Category Blocker: Inhibitor
Unit 50 mg
Description Unnatural fatty acid-neurotransmitter conjugate. Potent TRPV1 antagonist (IC50=40nM). Inhibits fatty acid amide hydrolase (FAAH) (IC50=5.6mM). Enhances levels of anandamide and 2-AG in vivo. Displays analgesic activity in both acute and chronic peripheral pain models but shows little efficacy in an inflammatory bowel disease model